CYM-5520
Product Name : CYM-5520Description:CYM-5520 is a selective and allosteric sphingosine 1-phosphate receptor 2 (S1PR2) agonist with an EC50 of 480 nM. CYM-5520 does not activate S1PR1, S1PR3, S1PR4 and S1PR5…
December 2024
CP-609754
Product Name : CP-609754Description:CP-609754 (LNK-754) is a potent and reversible farnesyltransferase inhibitor with potential anticancer activity.The IC50 for inhibiting farnesylation of recombinant human H-Ras is 0.57 ng/mL and recombinant K-Ras…
SMARCA-BD ligand 1 for Protac
Product Name : SMARCA-BD ligand 1 for ProtacDescription:SMARCA-BD ligand 1 for Protac is a compound that binds to the BAF ATPase subunits SMARCA2, and used for degrading SMARCA2, based on…
Obatoclax
Product Name : ObatoclaxDescription:Obatoclax (GX15-070), a BH3 mimetic, is a pan-BCL-2 family proteins inhibitor with a Ki of 220 nM for BCL-2. Obatoclax induces autophagy-dependent cell death and targets cyclin…
PSMA-11 free base
Product Name : PSMA-11 free baseDescription:PSMA-11, also known as DKFZ-PSMA-11, HBED-CC-PSMA or Psma-hbed-CC, is a ligand to make gallium Ga 68-labeled PSMA-11, which has potential use as a tracer for…
Copanlisib dihydrochloride
Product Name : Copanlisib dihydrochlorideDescription:Copanlisib dihydrochloride (BAY 80-6946 dihydrochloride) is a potent, selective and ATP-competitive pan-class I PI3K inhibitor, with IC50s of 0.5 nM, 0.7 nM, 3.7 nM and 6.4…
Benzoylgomisin P
Product Name : Benzoylgomisin PDescription:Benzoylgomisin P is an anti-inflammatory agent.CAS: 129445-43-8Molecular Weight:536.57Formula: C30H32O9Chemical Name: 9-hydroxy-3, 4, 5, 19-tetramethoxy-9, 10-dimethyl-15, 17-dioxatetracyclononadeca-1(19), 2(7), 3, 5, 12, 14(18)-hexaen-8-yl benzoateSmiles : CC1CC2=CC3OCOC=3C(OC)=C2C2=C(C=C(OC)C(OC)=C2OC)C(OC(=O)C2C=CC=CC=2)C1(C)OInChiKey: UFCGDBKFOKKVAC-UHFFFAOYSA-NInChi :…
Tumulosic acid
Product Name : Tumulosic acidDescription:Tumulosic acid, a triterpenoid, inhibits KLK5 protease activity (IC50= 14.84 μM). Tumulosic acid suppresses the proteolytic processing of LL-37 in keratinocytes at ≤10 μM.CAS: 508-24-7Molecular Weight:486.73Formula:…
β-Secretase Inhibitor II
Product Name : β-Secretase Inhibitor IIDescription:β-Secretase Inhibitor II is a β-Secretase inhibitor. β-Secretase Inhibitor II is a simple tripeptide aldehyde (IC50=700 nM for inhibition of total Aβ and IC50=2.5 μM…
(R)-(4′-Hydroxy)-5, 7-dihydroxy-4-chromanone
Product Name : (R)-(4′-Hydroxy)-5, 7-dihydroxy-4-chromanoneDescription:(R)-(4′-Hydroxy)-5,7-dihydroxy-4-chromanone, a homoisoflavonoid, has antiangiogenic activity against human retinal microvascular endothelial cells.CAS: 849727-88-4Molecular Weight:286.28Formula: C16H14O5Chemical Name: (3R)-5,7-dihydroxy-3--3,4-dihydro-2H-1-benzopyran-4-oneSmiles : OC1C=C(O)C2C(=O)(CC3C=CC(O)=CC=3)COC=2C=1InChiKey: FIASLUPJXGTCKM-SNVBAGLBSA-NInChi : InChI=1S/C16H14O5/c17-11-3-1-9(2-4-11)5-10-8-21-14-7-12(18)6-13(19)15(14)16(10)20/h1-4,6-7,10,17-19H,5,8H2/t10-/m1/s1Purity: ≥98% (or refer to…